Schedules of Controlled Substances: Placement of cyclopentyl fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl fentanyl in Schedule I, 75231-75235 [2020-22757]
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Federal Register / Vol. 85, No. 228 / Wednesday, November 25, 2020 / Rules and Regulations
For the Nuclear Regulatory Commission.
Pamela J. Shepherd-Vladimir,
Acting Chief Regulatory Analysis and
Rulemaking Support Branch, Division of
Rulemaking, Environmental, and Financial
Support, Office of Nuclear Material Safety
and Safeguards.
Control Division, Drug Enforcement
Administration; Mailing Address: 8701
Morrissette Drive, Springfield, Virginia
22152; Telephone: (571) 362–3261.
SUPPLEMENTARY INFORMATION:
[FR Doc. 2020–25875 Filed 11–24–20; 8:45 am]
BILLING CODE 7590–01–P
DEPARTMENT OF JUSTICE
Drug Enforcement Administration
21 CFR Part 1308
[Docket No. DEA–565]
Schedules of Controlled Substances:
Placement of cyclopentyl fentanyl,
isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl in Schedule I
Drug Enforcement
Administration, Department of Justice.
ACTION: Final rule.
AGENCY:
The Drug Enforcement
Administration places cyclopentyl
fentanyl (N-(1-phenethylpiperidin-4-yl)N-phenylcyclopentanecarboxamide),
isobutyryl fentanyl (N-(1phenethylpiperidin-4-yl)-Nphenylisobutyramide), parachloroisobutyryl fentanyl (N-(4chlorophenyl)-N-(1-phenethylpiperidin4-yl)isobutyramide), paramethoxybutyryl fentanyl (N-(4methoxyphenyl)-N-(1phenethylpiperidin-4-yl)butyramide),
and valeryl fentanyl (N-(1phenethylpiperidin-4-yl)-Nphenylpentanamide), including their
isomers, esters, ethers, salts, and salts of
isomers, esters, and ethers whenever the
existence of such isomers, esters, ethers,
and salts is possible, in schedule I of the
Controlled Substances Act. This action
continues the imposition of the
regulatory controls and administrative,
civil, and criminal sanctions applicable
to schedule I controlled substances on
persons who handle (manufacture,
distribute, import, export, engage in
research, conduct instructional
activities or chemical analysis with, or
possess), or propose to handle
cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl.
DATES: Effective date: November 25,
2020.
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SUMMARY:
FOR FURTHER INFORMATION CONTACT:
Scott A. Brinks, Regulatory Drafting and
Policy Support Section, Diversion
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Legal Authority
The Controlled Substances Act (CSA)
provides that proceedings for the
issuance, amendment, or repeal of the
scheduling of any drug or other
substance may be initiated by the
Attorney General (1) on his own motion;
(2) at the request of the Secretary of the
Department of Health and Human
Services (HHS); 1 or (3) on the petition
of any interested party. 21 U.S.C. 811(a).
This action was initiated on the
Attorney General’s own motion, as
delegated to the Administrator of DEA
(Administrator), and is supported by,
inter alia, a recommendation from the
Assistant Secretary for Health of HHS
(Assistant Secretary) and an evaluation
of all relevant data by the Drug
Enforcement Administration (DEA).
This action continues the imposition of
the regulatory controls and
administrative, civil, and criminal
sanctions of schedule I controlled
substances on any person who handles
or proposes to handle cyclopentyl
fentanyl, isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl.
Background
On February 1, 2018, DEA published
an order in the Federal Register
amending 21 CFR 1308.11(h) to
temporarily place cyclopentyl fentanyl
(N-(1-phenethylpiperidin-4-yl)-Nphenylcyclopentanecarboxamide),
isobutyryl fentanyl (N-(1phenethylpiperidin-4-yl)-Nphenylisobutyramide), parachloroisobutyryl fentanyl (N-(4chlorophenyl)-N-(1-phenethylpiperidin4-yl)isobutyramide), paramethoxybutyryl fentanyl (N-(4methoxyphenyl)-N-(1phenethylpiperidin-4-yl)butyramide),
and valeryl fentanyl (N-(1phenethylpiperidin-4-yl)-Nphenylpentanamide), along with two
other substances,2 in schedule I of the
1 As discussed in a memorandum of
understanding entered into by the Food and Drug
Administration (FDA) and the National Institute on
Drug Abuse (NIDA), FDA acts as the lead agency
within HHS in carrying out the Secretary’s
scheduling responsibilities under the CSA, with the
concurrence of NIDA. 50 FR 9518, Mar. 8, 1985.
The Secretary of HHS has delegated to the Assistant
Secretary for Health of HHS the authority to make
domestic drug scheduling recommendations. 58 FR
35460, July 1, 1993.
2 Those two other substances, ocfentanil (N-(2fluorophenyl)-2-methoxy-N-(phenethylpiperidin-4-
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75231
CSA pursuant to the temporary
scheduling provisions of 21 U.S.C.
811(h). 83 FR 4580. That temporary
scheduling order was effective on the
date of publication, and was based on
findings by the former Acting
Administrator that the temporary
scheduling of these seven substances
was necessary to avoid an imminent
hazard to the public safety pursuant to
21 U.S.C. 811(h)(1). On January 30,
2020, DEA published an order to extend
the temporary schedule I status of
cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl by one year, or
until February 1, 2021, pursuant to 21
CFR 811(h)(2). 85 FR 5321. Also, on that
same date and in the same issue of the
Federal Register, DEA simultaneously
published a notice of proposed
rulemaking (NPRM) to permanently
control cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl in schedule I of the
CSA. 85 FR 5356. Specifically, DEA
proposed to add these five substances to
the opiates list under 21 CFR
1308.11(b).
DEA and HHS Eight Factor Analyses
On November 12, 2019, the Assistant
Secretary submitted HHS’s scientific
and medical evaluation and scheduling
recommendation for cyclopropyl
fentanyl, para-fluorobutyryl fentanyl,
cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl to the former
Acting Administrator.3 After
considering the eight factors in 21
U.S.C. 811(c), each substance’s abuse
potential, lack of legitimate medical use
in the United States, and lack of
accepted safety for use under medical
supervision pursuant to 21 U.S.C.
812(b), the Assistant Secretary
recommended that cyclopentyl fentanyl,
isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl be controlled in schedule I of
the CSA. In response, DEA conducted
its own eight-factor analysis of
cyclopentyl fentanyl, isobutyryl
yl)acetamide) and para-fluorobutyryl fentanyl (N(4-fluorophenyl)-N-(1-phenethylpiperidin-4yl)butyramide, were subsequently permanently
placed in schedule I on November 29, 2018 (83 FR
61320) and October 25, 2019 (84 FR 57323),
respectively, pursuant to 21 U.S.C. 811(d)(1).
3 Although HHS also provided information on
cyclopropyl fentanyl and para-fluorobutyryl
fentanyl, these two substances will not be discussed
in this final rule since they were permanently
placed in schedule I on October 25, 2019. 84 FR
57323.
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fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl. DEA and HHS
analyses are available in their entirety in
the public docket for this rule (Docket
Number DEA–565) at https://
www.regulations.gov under ‘‘Supporting
Documents.’’
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Determination To Schedule cyclopentyl
fentanyl, isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl
After a review of the available data,
including the scientific and medical
evaluation and the scheduling
recommendations from HHS, DEA
published an NPRM entitled ‘‘Schedules
of Controlled Substances: Placement of
cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl into schedule I.’’
This rule proposed to control
cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl, including their
isomers, esters, ethers, salts, and salts of
isomers, esters, and ethers whenever the
existence of such isomers, esters, ethers,
and salts is possible, in schedule I of the
CSA. 85 FR 5356, January 30, 2020. The
NPRM provided an opportunity for
interested persons to file a request for
hearing in accordance with DEA
regulations on or before March 2, 2020.
No requests for such a hearing were
received by DEA. The NPRM also
provided an opportunity for interested
persons to submit comments on or
before March 2, 2020.
Comments Received
DEA received six comments on the
proposed rule to permanently control
cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl in schedule I of the
CSA. The submissions were from
individual or anonymous commenters.
Two commenters provided support for
the rule, and one commenter opposed
the rule. Three other commenters either
supported or opposed the proposal, but
misunderstood it to be rescheduling
fentanyl from schedule II to schedule I.
As such, the latter three comments were
outside the scope of this current
scheduling action.
Comment: The two commenters
provided different reasons for
supporting the proposed rule. One
commenter stated the proposed rule was
beneficial and expressed displeasure
with drug dealers, but did not elaborate
further. The other commenter stated that
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according to the Centers for Disease
Control and Prevention, abusing
unregulated opioids represents a
significant risk of opioid overdose to
users. Additionally, the commenter
stated that the opioid abuse epidemic is
incurring not only financial, but also
social and emotional damage. Lastly,
this commenter stated that these five
substances meet DEA’s requirements for
schedule I control, and noted they are
structurally similar to the opioid
fentanyl, lack FDA approval for
treatment, and are of unknown quality
and potency.
DEA Response: DEA appreciates the
comments in support of this
rulemaking.
Comment: One commenter stated that
DEA’s proposal to only place five
structural variants of fentanyl in
schedule I is ‘‘stupid’’ and will not solve
the problem when ‘‘China imports [sic]
four hundred variants’’ (taken to be
asserting that China exports 400 such
variants of fentanyl to the United
States). The commenter suggested that
DEA determine every possible ‘‘fentanyl
variant’’ and place them all in schedule
I rather than control individual
substances.
DEA Response: Similar to what this
commenter suggested, the agency has
undertaken a broad scheduling action
for fentanyl-related substances.
Specifically, on February 6, 2018, the
former Acting Administrator of DEA
published an order to temporarily
schedule fentanyl-related substances, a
class of substances as defined in the
order, and their isomers, esters, ethers,
salts, and salts of isomers, esters, and
ethers in schedule I. 83 FR 5188. This
temporary order defined a fentanylrelated substance to mean any substance
not otherwise controlled in any
schedule (i.e., not listed under another
DEA Controlled Substance Code
Number), and for which no exemption
or approval is in effect under section
505 of the Federal Food, Drug, and
Cosmetic Act (21 U.S.C. 355), that is
structurally related to fentanyl by one or
more of five specified structural
modifications. The class of fentanylrelated substances that was the subject
of the February 6, 2018, temporary
scheduling order is currently listed in
21 CFR 1308.11(h)(30). Although the
temporary scheduling of the fentanylrelated substances was scheduled to
expire on February 6, 2020, Congress
enacted a new law to extend the
temporary scheduling of all of those
fentanyl-related substances until May 6,
2021. (Pub. L. 116–114, Sec. 2).
As indicated above, the final rule
being issued today applies to five
fentanyl-related substances that were
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the subject of a February 1, 2018
temporary scheduling order (which was
issued five days prior to the class-wide
temporary scheduling of fentanylrelated substances). These five
substances will now be listed in 21 CFR
1308.11(b), as specified in the text of the
rule that appears below.
Scheduling Conclusion
After consideration of the relevant
matter presented through public
comments, the scientific and medical
evaluation and accompanying
recommendation of HHS, and after its
own eight-factor evaluation, DEA finds
that these facts and all other relevant
data constitute substantial evidence of
the potential for abuse of cyclopentyl
fentanyl, isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl. DEA is permanently
scheduling cyclopentyl fentanyl,
isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl as schedule I controlled
substances under the CSA.
Determination of Appropriate Schedule
The CSA establishes five schedules of
controlled substances known as
schedules I, II, III, IV, and V. The CSA
also specifies the findings required to
place a drug or other substance in any
particular schedule. 21 U.S.C. 812(b).
After consideration of the analysis and
recommendation of the Assistant
Secretary for HHS and review of all
other available data, the Acting
Administrator of DEA, pursuant to 21
U.S.C. 811(a) and 812(b)(1), finds the
following:
(1) The abuse potential of cyclopentyl
fentanyl, isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl is associated with each
substance’s pharmacological similarity
to other schedule I and II mu-opioid
receptor agonist substances which have
a high potential for abuse. Similar to
morphine (schedule II), fentanyl
(schedule II), and several schedule I
opioid substances that are structurally
related to fentanyl, cyclopentyl fentanyl,
isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl have been shown to bind and
act as mu-opioid receptor agonists;
(2) Cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl have no currently
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accepted medical use in treatment in the
United States; 4 and
(3) There is a lack of accepted safety
for use of cyclopentyl fentanyl,
isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl under medical supervision.
Based on these findings, the Acting
Administrator of DEA concludes that
cyclopentyl fentanyl (N-(1phenethylpiperidin-4-yl)-Nphenylcyclopentanecarboxamide),
isobutyryl fentanyl (N-(1phenethylpiperidin-4-yl)-Nphenylisobutyramide), parachloroisobutyryl fentanyl (N-(4chlorophenyl)-N-(1-phenethylpiperidin4-yl)isobutyramide), paramethoxybutyryl fentanyl (N-(4methoxyphenyl)-N-(1phenethylpiperidin-4-yl)butyramide),
and valeryl fentanyl (N-(1phenethylpiperidin-4-yl)-Nphenylpentanamide), including their
isomers, esters, ethers, salts, and salts of
isomers, esters, and ethers whenever the
existence of such isomers, esters, ethers,
and salts is possible, warrant control in
schedule I of the CSA. 21 U.S.C.
812(b)(1).
This final rule does not affect the
scheduling of fentanyl itself, which
remains a Schedule II controlled
substance.
Requirements for Handling cyclopentyl
fentanyl, isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl
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Cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl will continue 5 to
4 Although there is no evidence suggesting that
cyclopentyl fentanyl, isobutyryl fentanyl, parachloroisobutyryl fentanyl, para-methoxybutyryl
fentanyl, and valeryl fentanyl have a currently
accepted medical use in treatment in the United
States, it bears noting that a drug cannot be found
to have such medical use unless DEA concludes
that it satisfies a five-part test. Specifically, with
respect to a drug that has not been approved by
FDA, to have a currently accepted medical use in
treatment in the United States, all of the following
must be demonstrated:
i. The drug’s chemistry must be known and
reproducible;
ii. there must be adequate safety studies;
iii. there must be adequate and well-controlled
studies proving efficacy;
iv. the drug must be accepted by qualified
experts; and
v. the scientific evidence must be widely
available.
57 FR 10499 (1992).
5 Cyclopentyl fentanyl, isobutyryl fentanyl, parachloroisobutyryl fentanyl, para-methoxybutyryl
fentanyl, and valeryl fentanyl have been subject to
schedule I controls on a temporary basis, pursuant
to 21 U.S.C. 811(h), by virtue of the February 1,
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be subject to the CSA’s schedule I
regulatory controls and administrative,
civil, and criminal sanctions applicable
to the manufacture, distribution,
dispensing, importing, exporting,
research, and conduct of instructional
activities, including the following:
1. Registration. Any person who
handles (manufactures, distributes,
dispenses, imports, exports, engages in
research, or conducts instructional
activities or chemical analysis with, or
possesses) cyclopentyl fentanyl,
isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl, or who desires to handle
cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl, is required to be
registered with DEA to conduct such
activities pursuant to 21 U.S.C. 822,
823, 957, and 958, and in accordance
with 21 CFR parts 1301 and 1312.
2. Security. Cyclopentyl fentanyl,
isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl are subject to schedule I
security requirements and must be
handled and stored pursuant to 21
U.S.C. 821, 823, and in accordance with
21 CFR 1301.71–1301.93. Nonpractitioners handling these five
substances must also comply with the
employee screening requirements of 21
CFR 1301.90–1301.93.
3. Labeling and Packaging. All labels
and labeling for commercial containers
of cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl must be in
compliance with 21 U.S.C. 825 and
958(e), and be in accordance with 21
CFR part 1302.
4. Quota. Only registered
manufacturers are permitted to
manufacture cyclopentyl fentanyl,
isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl in accordance with a quota
assigned pursuant to 21 U.S.C. 826 and
in accordance with 21 CFR part 1303.
5. Inventory. Any person registered
with DEA to handle cyclopentyl
fentanyl, isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl must have an initial inventory
of all stocks of controlled substances
(including these substances) on hand on
the date the registrant first engages in
2018 temporary scheduling order (83 FR 4580) and
the subsequent one-year extension of that order
(January 30, 2020, 85 FR 5321).
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75233
the handling of controlled substances
pursuant to 21 U.S.C. 827 and 958, and
in accordance with 21 CFR 1304.03,
1304.04, and 1304.11.
After the initial inventory, every DEA
registrant must take a new inventory of
all stocks of controlled substances
(including cyclopentyl fentanyl,
isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl) on hand every two years
pursuant to 21 U.S.C. 827 and 958, and
in accordance with 21 CFR 1304.03,
1304.04, and 1304.11.
6. Records and Reports. Every DEA
registrant is required to maintain
records and submit reports with respect
to cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl, pursuant to 21
U.S.C. 827 and 958(e), and in
accordance with 21 CFR parts 1304 and
1312.
7. Order Forms. Every DEA registrant
who distributes cyclopentyl fentanyl,
isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl is required to comply with the
order form requirements, pursuant to 21
U.S.C. 828, and 21 CFR part 1305.
8. Importation and Exportation. All
importation and exportation of
cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl must be in
compliance with 21 U.S.C. 952, 953,
957, and 958, and in accordance with 21
CFR part 1312.
9. Liability. Any activity involving
cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl not authorized by,
or in violation of, the CSA or its
implementing regulations is unlawful,
and may subject the person to
administrative, civil, and/or criminal
sanctions.
Regulatory Analyses
Executive Orders (E.O.) 12866, 13563,
and 13771, Regulatory Planning and
Review, Improving Regulation and
Regulatory Review, and Reducing
Regulation and Controlling Regulatory
Costs
In accordance with 21 U.S.C. 811(a),
this final scheduling action is subject to
formal rulemaking procedures
performed ‘‘on the record after
opportunity for a hearing,’’ which are
conducted pursuant to the provisions of
5 U.S.C. 556 and 557. The CSA sets
forth the criteria for scheduling a drug
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or other substance. Such actions are
exempt from review by the Office of
Management and Budget (OMB)
pursuant to section 3(d)(1) of E.O. 12866
and the principles reaffirmed in E.O.
13563.
This final rule does not meet the
definition of an E.O. 13771 regulatory
action. OMB has previously determined
that formal rulemaking actions
concerning the scheduling of controlled
substances, such as this rule, are not
significant regulatory actions under
section 3(f) of E.O. 12866.
Executive Order 12988
This regulation meets the applicable
standards set forth in sections 3(a) and
3(b)(2) of E.O. 12988 to eliminate
drafting errors and ambiguity, minimize
litigation, provide a clear legal standard
for affected conduct, and promote
simplification and burden reduction.
Executive Order 13132
This rulemaking does not have
federalism implications warranting the
application of E.O. 13132. The rule does
not have substantial direct effects on the
States, on the relationship between the
national government and the States, or
the distribution of power and
responsibilities among the various
levels of government.
Executive Order 13175
This rule does not have tribal
implications warranting the application
of E.O. 13175. It does not have
substantial direct effects on one or more
Indian tribes, on the relationship
between the Federal government and
Indian tribes, or on the distribution of
power and responsibilities between the
Federal government and Indian tribes.
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Regulatory Flexibility Act
The Acting Administrator, in
accordance with the Regulatory
Flexibility Act (RFA), 5 U.S.C. 601–602,
has reviewed this final rule and, by
approving it, certifies that it will not
have a significant economic impact on
a substantial number of small entities.
On February 1, 2018, DEA published an
order to temporarily place cyclopentyl
fentanyl, isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl in schedule I of the CSA
pursuant to the temporary scheduling
provisions of 21 U.S.C. 811(h). DEA
estimates that all entities handling or
planning to handle cyclopentyl
fentanyl, isobutyryl fentanyl, parachloroisobutyryl fentanyl, paramethoxybutyryl fentanyl, and valeryl
fentanyl have already established and
implemented the systems and processes
required to handle these substances.
As discussed in the NPRM, there are
34 registrations authorized to handle
one or more of the following substances:
cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
or valeryl fentanyl, as well as a number
of registered analytical labs that are
authorized to handle schedule I
controlled substances generally. These
34 registrations represent 26 entities, of
which eight are small entities.
Therefore, DEA estimates eight small
entities are affected by this rule.
A review of the 34 registrations
indicates that all entities that currently
handle cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl also handle other
schedule I controlled substances and
have established and implemented (or
maintain) the systems and processes
required to handle these substances.
Therefore, DEA anticipates that this
final rule will impose minimal or no
economic impact on any affected
entities, and, thus, will not have a
significant economic impact on any of
the eight affected small entities.
Therefore, DEA has concluded that this
final rule will not have a significant
economic impact on a substantial
number of small entities.
Unfunded Mandates Reform Act of 1995
In accordance with the Unfunded
Mandates Reform Act (UMRA) of 1995,
2 U.S.C. 1501 et seq., DEA has
determined and certifies that this action
would not result in any Federal
mandate that may result ‘‘in the
expenditure by State, local, and tribal
governments, in the aggregate, or by the
private sector, of $100 million or more
(adjusted annually for inflation) in any
1 year * * * .’’ Therefore, neither a
Small Government Agency Plan nor any
other action is required under UMRA of
1995.
Paperwork Reduction Act of 1995
This action does not impose a new
collection of information under the
Paperwork Reduction Act of 1995. 44
U.S.C. 3501–3521. This action would
not impose recordkeeping or reporting
requirements on State or local
governments, individuals, businesses, or
organizations. An agency may not
conduct or sponsor, and a person is not
required to respond to, a collection of
information unless it displays a
currently valid OMB control number.
Congressional Review Act
This rule is not a major rule as
defined by the Congressional Review
Act (CRA), 5 U.S.C. 804. This rule will
not result in: ‘‘an annual effect on the
economy of $100 million or more; a
major increase in costs or prices for
consumers, individual industries,
Federal, State, or local government
agencies, or geographic regions; or
significant adverse effects on
competition, employment, investment,
productivity, innovation, or on the
ability of United States-based
enterprises to compete with foreignbased enterprises in domestic and
export markets.’’ However, pursuant to
the CRA, DEA has submitted a copy of
this final rule to both Houses of
Congress and to the Comptroller
General.
List of Subjects in 21 CFR Part 1308
Administrative practice and
procedure, Drug traffic control,
Reporting and recordkeeping
requirements.
For the reasons set out above, 21 CFR
part 1308 is amended as follows:
PART 1308—SCHEDULES OF
CONTROLLED SUBSTANCES
1. The authority citation for 21 CFR
part 1308 continues to read as follows:
■
Authority: 21 U.S.C. 811, 812, 871(b),
956(b), unless otherwise noted.
2. In § 1308.11:
a. Revise paragraphs (b)(22), (40), (56),
and (59);
■ b. Add paragraph (b)(75);
■ c. Remove and reserve paragraphs
(h)(23), and (h)(25) through (h)(28).
The revisions and addition read as
follows:
■
■
§ 1308.11
*
Schedule I.
*
*
(b) * * *
*
*
(22) Cyclopentyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N-phenylcyclopentanecarboxamide) ......................................................
9847
*
*
*
*
*
*
(40) Isobutyryl fentanyl (N-(1-phenethylpiperidin-4-yl)-N-phenylisobutyramide) ............................................................................
*
*
*
*
*
*
*
(56) para-Chloroisobutyryl fentanyl (N-(4-chlorophenyl)-N-(1-phenethylpiperidin-4-yl)isobutyramide .........................................
*
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Federal Register / Vol. 85, No. 228 / Wednesday, November 25, 2020 / Rules and Regulations
*
*
*
*
*
*
(59) para-Methoxybutyryl fentanyl (N-(4-methoxyphenyl)-N-(1-phenethylpiperidin-4-yl)butyramide) ..........................................
*
*
*
*
*
*
*
(75) Valeryl fentanyl (N-(1-phenethylpiperidin-4-yl)-N-phenylpentanamide) ...................................................................................
*
*
*
*
*
*
Timothy J. Shea,
Acting Administrator.
[FR Doc. 2020–22757 Filed 11–24–20; 8:45 am]
BILLING CODE 4410–09–P
ENVIRONMENTAL PROTECTION
AGENCY
40 CFR Part 63
[EPA–HQ–OAR–2018–0747; FRL–10010–12–
OAR]
RIN 2060–AU16
National Emission Standards for
Hazardous Air Pollutants:
Miscellaneous Coating Manufacturing
Residual Risk and Technology Review
Correction
In rule document 2020–13439
beginning on page 49724 in the issue of
August 14, 2020, make the following
correction:
§ 63.8000
[Corrected]
On page 49742, in the first column, in
§ 63.8000(vi), in the 14th line ‘‘August
15, 2022’’ should read ‘‘August 15,
2018’’.
■
[FR Doc. C1–2020–13439 Filed 11–24–20; 8:45 am]
BILLING CODE 1301–00–D
ENVIRONMENTAL PROTECTION
AGENCY
40 CFR Part 711
[EPA–HQ–OPPT–2018–0321; FRL–10016–
96]
RIN 2070–AK33
Chemical Data Reporting; Final
Extension of the 2020 Submission
Period
Environmental Protection
Agency (EPA).
ACTION: Final rule.
AGENCY:
The Environmental Protection
Agency (EPA) is amending the Toxic
Substances Control Act (TSCA)
Chemical Data Reporting (CDR)
regulations by extending the submission
deadline for 2020 reports to January 29,
2021. This is the final extension for the
2020 submission period only. The CDR
SUMMARY:
jbell on DSKJLSW7X2PROD with RULES
75235
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regulations require manufacturers
(including importers) of certain
chemical substances included on the
TSCA Chemical Substance Inventory
(TSCA Inventory) to report data on the
manufacturing, processing, and use of
the chemical substances.
DATES: This final rule is effective
November 25, 2020.
ADDRESSES: The docket for this action,
identified by docket identification (ID)
number EPA–HQ–OPPT–2018–0321, is
available at https://www.regulations.gov
or at the Office of Pollution Prevention
and Toxics Docket (OPPT Docket),
Environmental Protection Agency
Docket Center (EPA/DC), West, William
Jefferson Clinton Bldg., Rm. 3334, 1301
Constitution Ave. NW, Washington, DC.
The Public Reading Room is open from
8:30 a.m. to 4:30 p.m., Monday through
Friday, excluding legal holidays. The
telephone number for the Public
Reading Room is (202) 566–1744, and
the telephone number for the OPPT
Docket is (202) 566–0280.
Please note that due to the public
health emergency the EPA Docket
Center (EPA/DC) and Reading Room
was closed to public visitors on March
31, 2020. Our EPA/DC staff will
continue to provide customer service
via email, phone, and webform. For
further information on EPA/DC services,
docket contact information and the
current status of the EPA/DC and
Reading Room, please visit https://
www.epa.gov/dockets.
FOR FURTHER INFORMATION CONTACT: For
technical information contact: Susan
Sharkey, Data Gathering and Analysis
Division (7406M), Office of Pollution
Prevention and Toxics, Environmental
Protection Agency, 1200 Pennsylvania
Ave. NW, Washington, DC 20460–0001;
telephone number: (202) 564–8789;
email address: sharkey.susan@epa.gov.
For general information contact: The
TSCA-Hotline, ABVI-Goodwill, 422
South Clinton Ave., Rochester, NY
14620; telephone number: (202) 554–
1404; email address: TSCA-Hotline@
epa.gov.
SUPPLEMENTARY INFORMATION:
I. General Information
A. Does this action apply to me?
You may be potentially affected by
this action if you manufacture
(including import) chemical substances
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9840
listed on the TSCA Inventory. The
following list of North American
Industrial Classification System
(NAICS) codes is not intended to be
exhaustive, but rather provides a guide
to help readers determine whether this
document applies to them. Potentially
affected entities may include but are not
limited to:
• Chemical manufacturers (including
importers) (NAICS codes 325 and
324110, e.g., chemical manufacturing
and processing and petroleum
refineries).
• Chemical users and processors who
may manufacture a byproduct chemical
substance (NAICS codes 22, 322, 331,
and 3344, e.g., utilities, paper
manufacturing, primary metal
manufacturing, and semiconductor and
other electronic component
manufacturing).
B. What action is the Agency taking?
The current 2020 CDR submission
period is from June 1 to November 30,
2020 (on April 9, 2020, EPA extended
the September 30, 2020 deadline to
November 30, 2020 (see 85 FR 19890)).
EPA is issuing this amendment to
extend the deadline for 2020 CDR
submission reports until January 29,
2021. This is an extension for the 2020
submission period only: Subsequent
submission periods (recurring every
four years, next in 2024) are not being
amended.
The Agency is taking this action in
response to concerns raised by the
regulated community about their ability
to submit the required information
within the prescribed period. Written
requests to extend the CDR submission
period have been received by the
Agency starting in late-September.
Copies of these letters are included in
the docket (see ADDRESSES), and, at the
time of drafting this document, include
the following specific communications:
• Air Products and Chemicals, Inc.
2020 CDR 90-day Extension Request
[Letter]. September 25, 2020. Certain
information needed to inform
submissions is stored off-site and
reviewing in-person presents a logistical
challenge because of the COVID–19
pandemic (administrative staff is
currently on business-critical or work
from home status). (Ref. 1.)
• American Chemistry Council
(ACC). Request for an Extension to the
TSCA Chemical Data Reporting (CDR)
E:\FR\FM\25NOR1.SGM
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Agencies
[Federal Register Volume 85, Number 228 (Wednesday, November 25, 2020)]
[Rules and Regulations]
[Pages 75231-75235]
From the Federal Register Online via the Government Publishing Office [www.gpo.gov]
[FR Doc No: 2020-22757]
=======================================================================
-----------------------------------------------------------------------
DEPARTMENT OF JUSTICE
Drug Enforcement Administration
21 CFR Part 1308
[Docket No. DEA-565]
Schedules of Controlled Substances: Placement of cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl in Schedule I
AGENCY: Drug Enforcement Administration, Department of Justice.
ACTION: Final rule.
-----------------------------------------------------------------------
SUMMARY: The Drug Enforcement Administration places cyclopentyl
fentanyl (N-(1-phenethylpiperidin-4-yl)-N-
phenylcyclopentanecarboxamide), isobutyryl fentanyl (N-(1-
phenethylpiperidin-4-yl)-N-phenylisobutyramide), para-chloroisobutyryl
fentanyl (N-(4-chlorophenyl)-N-(1-phenethylpiperidin-4-
yl)isobutyramide), para-methoxybutyryl fentanyl (N-(4-methoxyphenyl)-N-
(1-phenethylpiperidin-4-yl)butyramide), and valeryl fentanyl (N-(1-
phenethylpiperidin-4-yl)-N-phenylpentanamide), including their isomers,
esters, ethers, salts, and salts of isomers, esters, and ethers
whenever the existence of such isomers, esters, ethers, and salts is
possible, in schedule I of the Controlled Substances Act. This action
continues the imposition of the regulatory controls and administrative,
civil, and criminal sanctions applicable to schedule I controlled
substances on persons who handle (manufacture, distribute, import,
export, engage in research, conduct instructional activities or
chemical analysis with, or possess), or propose to handle cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl.
DATES: Effective date: November 25, 2020.
FOR FURTHER INFORMATION CONTACT: Scott A. Brinks, Regulatory Drafting
and Policy Support Section, Diversion Control Division, Drug
Enforcement Administration; Mailing Address: 8701 Morrissette Drive,
Springfield, Virginia 22152; Telephone: (571) 362-3261.
SUPPLEMENTARY INFORMATION:
Legal Authority
The Controlled Substances Act (CSA) provides that proceedings for
the issuance, amendment, or repeal of the scheduling of any drug or
other substance may be initiated by the Attorney General (1) on his own
motion; (2) at the request of the Secretary of the Department of Health
and Human Services (HHS); \1\ or (3) on the petition of any interested
party. 21 U.S.C. 811(a). This action was initiated on the Attorney
General's own motion, as delegated to the Administrator of DEA
(Administrator), and is supported by, inter alia, a recommendation from
the Assistant Secretary for Health of HHS (Assistant Secretary) and an
evaluation of all relevant data by the Drug Enforcement Administration
(DEA). This action continues the imposition of the regulatory controls
and administrative, civil, and criminal sanctions of schedule I
controlled substances on any person who handles or proposes to handle
cyclopentyl fentanyl, isobutyryl fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl, and valeryl fentanyl.
---------------------------------------------------------------------------
\1\ As discussed in a memorandum of understanding entered into
by the Food and Drug Administration (FDA) and the National Institute
on Drug Abuse (NIDA), FDA acts as the lead agency within HHS in
carrying out the Secretary's scheduling responsibilities under the
CSA, with the concurrence of NIDA. 50 FR 9518, Mar. 8, 1985. The
Secretary of HHS has delegated to the Assistant Secretary for Health
of HHS the authority to make domestic drug scheduling
recommendations. 58 FR 35460, July 1, 1993.
---------------------------------------------------------------------------
Background
On February 1, 2018, DEA published an order in the Federal Register
amending 21 CFR 1308.11(h) to temporarily place cyclopentyl fentanyl
(N-(1-phenethylpiperidin-4-yl)-N-phenylcyclopentanecarboxamide),
isobutyryl fentanyl (N-(1-phenethylpiperidin-4-yl)-N-
phenylisobutyramide), para-chloroisobutyryl fentanyl (N-(4-
chlorophenyl)-N-(1-phenethylpiperidin-4-yl)isobutyramide), para-
methoxybutyryl fentanyl (N-(4-methoxyphenyl)-N-(1-phenethylpiperidin-4-
yl)butyramide), and valeryl fentanyl (N-(1-phenethylpiperidin-4-yl)-N-
phenylpentanamide), along with two other substances,\2\ in schedule I
of the CSA pursuant to the temporary scheduling provisions of 21 U.S.C.
811(h). 83 FR 4580. That temporary scheduling order was effective on
the date of publication, and was based on findings by the former Acting
Administrator that the temporary scheduling of these seven substances
was necessary to avoid an imminent hazard to the public safety pursuant
to 21 U.S.C. 811(h)(1). On January 30, 2020, DEA published an order to
extend the temporary schedule I status of cyclopentyl fentanyl,
isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl by one year, or until
February 1, 2021, pursuant to 21 CFR 811(h)(2). 85 FR 5321. Also, on
that same date and in the same issue of the Federal Register, DEA
simultaneously published a notice of proposed rulemaking (NPRM) to
permanently control cyclopentyl fentanyl, isobutyryl fentanyl, para-
chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl
fentanyl in schedule I of the CSA. 85 FR 5356. Specifically, DEA
proposed to add these five substances to the opiates list under 21 CFR
1308.11(b).
---------------------------------------------------------------------------
\2\ Those two other substances, ocfentanil (N-(2-fluorophenyl)-
2-methoxy-N-(phenethylpiperidin-4-yl)acetamide) and para-
fluorobutyryl fentanyl (N-(4-fluorophenyl)-N-(1-phenethylpiperidin-
4-yl)butyramide, were subsequently permanently placed in schedule I
on November 29, 2018 (83 FR 61320) and October 25, 2019 (84 FR
57323), respectively, pursuant to 21 U.S.C. 811(d)(1).
---------------------------------------------------------------------------
DEA and HHS Eight Factor Analyses
On November 12, 2019, the Assistant Secretary submitted HHS's
scientific and medical evaluation and scheduling recommendation for
cyclopropyl fentanyl, para-fluorobutyryl fentanyl, cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl to the former Acting
Administrator.\3\ After considering the eight factors in 21 U.S.C.
811(c), each substance's abuse potential, lack of legitimate medical
use in the United States, and lack of accepted safety for use under
medical supervision pursuant to 21 U.S.C. 812(b), the Assistant
Secretary recommended that cyclopentyl fentanyl, isobutyryl fentanyl,
para-chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and
valeryl fentanyl be controlled in schedule I of the CSA. In response,
DEA conducted its own eight-factor analysis of cyclopentyl fentanyl,
isobutyryl
[[Page 75232]]
fentanyl, para-chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl. DEA and HHS analyses are available in their
entirety in the public docket for this rule (Docket Number DEA-565) at
https://www.regulations.gov under ``Supporting Documents.''
---------------------------------------------------------------------------
\3\ Although HHS also provided information on cyclopropyl
fentanyl and para-fluorobutyryl fentanyl, these two substances will
not be discussed in this final rule since they were permanently
placed in schedule I on October 25, 2019. 84 FR 57323.
---------------------------------------------------------------------------
Determination To Schedule cyclopentyl fentanyl, isobutyryl fentanyl,
para-chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and
valeryl fentanyl
After a review of the available data, including the scientific and
medical evaluation and the scheduling recommendations from HHS, DEA
published an NPRM entitled ``Schedules of Controlled Substances:
Placement of cyclopentyl fentanyl, isobutyryl fentanyl, para-
chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl
fentanyl into schedule I.'' This rule proposed to control cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl, including their isomers,
esters, ethers, salts, and salts of isomers, esters, and ethers
whenever the existence of such isomers, esters, ethers, and salts is
possible, in schedule I of the CSA. 85 FR 5356, January 30, 2020. The
NPRM provided an opportunity for interested persons to file a request
for hearing in accordance with DEA regulations on or before March 2,
2020. No requests for such a hearing were received by DEA. The NPRM
also provided an opportunity for interested persons to submit comments
on or before March 2, 2020.
Comments Received
DEA received six comments on the proposed rule to permanently
control cyclopentyl fentanyl, isobutyryl fentanyl, para-
chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl
fentanyl in schedule I of the CSA. The submissions were from individual
or anonymous commenters. Two commenters provided support for the rule,
and one commenter opposed the rule. Three other commenters either
supported or opposed the proposal, but misunderstood it to be
rescheduling fentanyl from schedule II to schedule I. As such, the
latter three comments were outside the scope of this current scheduling
action.
Comment: The two commenters provided different reasons for
supporting the proposed rule. One commenter stated the proposed rule
was beneficial and expressed displeasure with drug dealers, but did not
elaborate further. The other commenter stated that according to the
Centers for Disease Control and Prevention, abusing unregulated opioids
represents a significant risk of opioid overdose to users.
Additionally, the commenter stated that the opioid abuse epidemic is
incurring not only financial, but also social and emotional damage.
Lastly, this commenter stated that these five substances meet DEA's
requirements for schedule I control, and noted they are structurally
similar to the opioid fentanyl, lack FDA approval for treatment, and
are of unknown quality and potency.
DEA Response: DEA appreciates the comments in support of this
rulemaking.
Comment: One commenter stated that DEA's proposal to only place
five structural variants of fentanyl in schedule I is ``stupid'' and
will not solve the problem when ``China imports [sic] four hundred
variants'' (taken to be asserting that China exports 400 such variants
of fentanyl to the United States). The commenter suggested that DEA
determine every possible ``fentanyl variant'' and place them all in
schedule I rather than control individual substances.
DEA Response: Similar to what this commenter suggested, the agency
has undertaken a broad scheduling action for fentanyl-related
substances. Specifically, on February 6, 2018, the former Acting
Administrator of DEA published an order to temporarily schedule
fentanyl-related substances, a class of substances as defined in the
order, and their isomers, esters, ethers, salts, and salts of isomers,
esters, and ethers in schedule I. 83 FR 5188. This temporary order
defined a fentanyl-related substance to mean any substance not
otherwise controlled in any schedule (i.e., not listed under another
DEA Controlled Substance Code Number), and for which no exemption or
approval is in effect under section 505 of the Federal Food, Drug, and
Cosmetic Act (21 U.S.C. 355), that is structurally related to fentanyl
by one or more of five specified structural modifications. The class of
fentanyl-related substances that was the subject of the February 6,
2018, temporary scheduling order is currently listed in 21 CFR
1308.11(h)(30). Although the temporary scheduling of the fentanyl-
related substances was scheduled to expire on February 6, 2020,
Congress enacted a new law to extend the temporary scheduling of all of
those fentanyl-related substances until May 6, 2021. (Pub. L. 116-114,
Sec. 2).
As indicated above, the final rule being issued today applies to
five fentanyl-related substances that were the subject of a February 1,
2018 temporary scheduling order (which was issued five days prior to
the class-wide temporary scheduling of fentanyl-related substances).
These five substances will now be listed in 21 CFR 1308.11(b), as
specified in the text of the rule that appears below.
Scheduling Conclusion
After consideration of the relevant matter presented through public
comments, the scientific and medical evaluation and accompanying
recommendation of HHS, and after its own eight-factor evaluation, DEA
finds that these facts and all other relevant data constitute
substantial evidence of the potential for abuse of cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl. DEA is permanently
scheduling cyclopentyl fentanyl, isobutyryl fentanyl, para-
chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl
fentanyl as schedule I controlled substances under the CSA.
Determination of Appropriate Schedule
The CSA establishes five schedules of controlled substances known
as schedules I, II, III, IV, and V. The CSA also specifies the findings
required to place a drug or other substance in any particular schedule.
21 U.S.C. 812(b). After consideration of the analysis and
recommendation of the Assistant Secretary for HHS and review of all
other available data, the Acting Administrator of DEA, pursuant to 21
U.S.C. 811(a) and 812(b)(1), finds the following:
(1) The abuse potential of cyclopentyl fentanyl, isobutyryl
fentanyl, para-chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl,
and valeryl fentanyl is associated with each substance's
pharmacological similarity to other schedule I and II mu-opioid
receptor agonist substances which have a high potential for abuse.
Similar to morphine (schedule II), fentanyl (schedule II), and several
schedule I opioid substances that are structurally related to fentanyl,
cyclopentyl fentanyl, isobutyryl fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl, and valeryl fentanyl have been
shown to bind and act as mu-opioid receptor agonists;
(2) Cyclopentyl fentanyl, isobutyryl fentanyl, para-
chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl
fentanyl have no currently
[[Page 75233]]
accepted medical use in treatment in the United States; \4\ and
---------------------------------------------------------------------------
\4\ Although there is no evidence suggesting that cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl have a currently
accepted medical use in treatment in the United States, it bears
noting that a drug cannot be found to have such medical use unless
DEA concludes that it satisfies a five-part test. Specifically, with
respect to a drug that has not been approved by FDA, to have a
currently accepted medical use in treatment in the United States,
all of the following must be demonstrated:
i. The drug's chemistry must be known and reproducible;
ii. there must be adequate safety studies;
iii. there must be adequate and well-controlled studies proving
efficacy;
iv. the drug must be accepted by qualified experts; and
v. the scientific evidence must be widely available.
57 FR 10499 (1992).
---------------------------------------------------------------------------
(3) There is a lack of accepted safety for use of cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl under medical
supervision.
Based on these findings, the Acting Administrator of DEA concludes
that cyclopentyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N-
phenylcyclopentanecarboxamide), isobutyryl fentanyl (N-(1-
phenethylpiperidin-4-yl)-N-phenylisobutyramide), para-chloroisobutyryl
fentanyl (N-(4-chlorophenyl)-N-(1-phenethylpiperidin-4-
yl)isobutyramide), para-methoxybutyryl fentanyl (N-(4-methoxyphenyl)-N-
(1-phenethylpiperidin-4-yl)butyramide), and valeryl fentanyl (N-(1-
phenethylpiperidin-4-yl)-N-phenylpentanamide), including their isomers,
esters, ethers, salts, and salts of isomers, esters, and ethers
whenever the existence of such isomers, esters, ethers, and salts is
possible, warrant control in schedule I of the CSA. 21 U.S.C.
812(b)(1).
This final rule does not affect the scheduling of fentanyl itself,
which remains a Schedule II controlled substance.
Requirements for Handling cyclopentyl fentanyl, isobutyryl fentanyl,
para-chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and
valeryl fentanyl
Cyclopentyl fentanyl, isobutyryl fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl, and valeryl fentanyl will
continue \5\ to be subject to the CSA's schedule I regulatory controls
and administrative, civil, and criminal sanctions applicable to the
manufacture, distribution, dispensing, importing, exporting, research,
and conduct of instructional activities, including the following:
---------------------------------------------------------------------------
\5\ Cyclopentyl fentanyl, isobutyryl fentanyl, para-
chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl
fentanyl have been subject to schedule I controls on a temporary
basis, pursuant to 21 U.S.C. 811(h), by virtue of the February 1,
2018 temporary scheduling order (83 FR 4580) and the subsequent one-
year extension of that order (January 30, 2020, 85 FR 5321).
---------------------------------------------------------------------------
1. Registration. Any person who handles (manufactures, distributes,
dispenses, imports, exports, engages in research, or conducts
instructional activities or chemical analysis with, or possesses)
cyclopentyl fentanyl, isobutyryl fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl, and valeryl fentanyl, or who
desires to handle cyclopentyl fentanyl, isobutyryl fentanyl, para-
chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl
fentanyl, is required to be registered with DEA to conduct such
activities pursuant to 21 U.S.C. 822, 823, 957, and 958, and in
accordance with 21 CFR parts 1301 and 1312.
2. Security. Cyclopentyl fentanyl, isobutyryl fentanyl, para-
chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl
fentanyl are subject to schedule I security requirements and must be
handled and stored pursuant to 21 U.S.C. 821, 823, and in accordance
with 21 CFR 1301.71-1301.93. Non-practitioners handling these five
substances must also comply with the employee screening requirements of
21 CFR 1301.90-1301.93.
3. Labeling and Packaging. All labels and labeling for commercial
containers of cyclopentyl fentanyl, isobutyryl fentanyl, para-
chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl
fentanyl must be in compliance with 21 U.S.C. 825 and 958(e), and be in
accordance with 21 CFR part 1302.
4. Quota. Only registered manufacturers are permitted to
manufacture cyclopentyl fentanyl, isobutyryl fentanyl, para-
chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl
fentanyl in accordance with a quota assigned pursuant to 21 U.S.C. 826
and in accordance with 21 CFR part 1303.
5. Inventory. Any person registered with DEA to handle cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl must have an initial
inventory of all stocks of controlled substances (including these
substances) on hand on the date the registrant first engages in the
handling of controlled substances pursuant to 21 U.S.C. 827 and 958,
and in accordance with 21 CFR 1304.03, 1304.04, and 1304.11.
After the initial inventory, every DEA registrant must take a new
inventory of all stocks of controlled substances (including cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl) on hand every two years
pursuant to 21 U.S.C. 827 and 958, and in accordance with 21 CFR
1304.03, 1304.04, and 1304.11.
6. Records and Reports. Every DEA registrant is required to
maintain records and submit reports with respect to cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl, pursuant to 21 U.S.C.
827 and 958(e), and in accordance with 21 CFR parts 1304 and 1312.
7. Order Forms. Every DEA registrant who distributes cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl is required to comply
with the order form requirements, pursuant to 21 U.S.C. 828, and 21 CFR
part 1305.
8. Importation and Exportation. All importation and exportation of
cyclopentyl fentanyl, isobutyryl fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl, and valeryl fentanyl must be in
compliance with 21 U.S.C. 952, 953, 957, and 958, and in accordance
with 21 CFR part 1312.
9. Liability. Any activity involving cyclopentyl fentanyl,
isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl not authorized by, or in
violation of, the CSA or its implementing regulations is unlawful, and
may subject the person to administrative, civil, and/or criminal
sanctions.
Regulatory Analyses
Executive Orders (E.O.) 12866, 13563, and 13771, Regulatory Planning
and Review, Improving Regulation and Regulatory Review, and Reducing
Regulation and Controlling Regulatory Costs
In accordance with 21 U.S.C. 811(a), this final scheduling action
is subject to formal rulemaking procedures performed ``on the record
after opportunity for a hearing,'' which are conducted pursuant to the
provisions of 5 U.S.C. 556 and 557. The CSA sets forth the criteria for
scheduling a drug
[[Page 75234]]
or other substance. Such actions are exempt from review by the Office
of Management and Budget (OMB) pursuant to section 3(d)(1) of E.O.
12866 and the principles reaffirmed in E.O. 13563.
This final rule does not meet the definition of an E.O. 13771
regulatory action. OMB has previously determined that formal rulemaking
actions concerning the scheduling of controlled substances, such as
this rule, are not significant regulatory actions under section 3(f) of
E.O. 12866.
Executive Order 12988
This regulation meets the applicable standards set forth in
sections 3(a) and 3(b)(2) of E.O. 12988 to eliminate drafting errors
and ambiguity, minimize litigation, provide a clear legal standard for
affected conduct, and promote simplification and burden reduction.
Executive Order 13132
This rulemaking does not have federalism implications warranting
the application of E.O. 13132. The rule does not have substantial
direct effects on the States, on the relationship between the national
government and the States, or the distribution of power and
responsibilities among the various levels of government.
Executive Order 13175
This rule does not have tribal implications warranting the
application of E.O. 13175. It does not have substantial direct effects
on one or more Indian tribes, on the relationship between the Federal
government and Indian tribes, or on the distribution of power and
responsibilities between the Federal government and Indian tribes.
Regulatory Flexibility Act
The Acting Administrator, in accordance with the Regulatory
Flexibility Act (RFA), 5 U.S.C. 601-602, has reviewed this final rule
and, by approving it, certifies that it will not have a significant
economic impact on a substantial number of small entities. On February
1, 2018, DEA published an order to temporarily place cyclopentyl
fentanyl, isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, and valeryl fentanyl in schedule I of the CSA
pursuant to the temporary scheduling provisions of 21 U.S.C. 811(h).
DEA estimates that all entities handling or planning to handle
cyclopentyl fentanyl, isobutyryl fentanyl, para-chloroisobutyryl
fentanyl, para-methoxybutyryl fentanyl, and valeryl fentanyl have
already established and implemented the systems and processes required
to handle these substances.
As discussed in the NPRM, there are 34 registrations authorized to
handle one or more of the following substances: cyclopentyl fentanyl,
isobutyryl fentanyl, para-chloroisobutyryl fentanyl, para-
methoxybutyryl fentanyl, or valeryl fentanyl, as well as a number of
registered analytical labs that are authorized to handle schedule I
controlled substances generally. These 34 registrations represent 26
entities, of which eight are small entities. Therefore, DEA estimates
eight small entities are affected by this rule.
A review of the 34 registrations indicates that all entities that
currently handle cyclopentyl fentanyl, isobutyryl fentanyl, para-
chloroisobutyryl fentanyl, para-methoxybutyryl fentanyl, and valeryl
fentanyl also handle other schedule I controlled substances and have
established and implemented (or maintain) the systems and processes
required to handle these substances. Therefore, DEA anticipates that
this final rule will impose minimal or no economic impact on any
affected entities, and, thus, will not have a significant economic
impact on any of the eight affected small entities. Therefore, DEA has
concluded that this final rule will not have a significant economic
impact on a substantial number of small entities.
Unfunded Mandates Reform Act of 1995
In accordance with the Unfunded Mandates Reform Act (UMRA) of 1995,
2 U.S.C. 1501 et seq., DEA has determined and certifies that this
action would not result in any Federal mandate that may result ``in the
expenditure by State, local, and tribal governments, in the aggregate,
or by the private sector, of $100 million or more (adjusted annually
for inflation) in any 1 year * * * .'' Therefore, neither a Small
Government Agency Plan nor any other action is required under UMRA of
1995.
Paperwork Reduction Act of 1995
This action does not impose a new collection of information under
the Paperwork Reduction Act of 1995. 44 U.S.C. 3501-3521. This action
would not impose recordkeeping or reporting requirements on State or
local governments, individuals, businesses, or organizations. An agency
may not conduct or sponsor, and a person is not required to respond to,
a collection of information unless it displays a currently valid OMB
control number.
Congressional Review Act
This rule is not a major rule as defined by the Congressional
Review Act (CRA), 5 U.S.C. 804. This rule will not result in: ``an
annual effect on the economy of $100 million or more; a major increase
in costs or prices for consumers, individual industries, Federal,
State, or local government agencies, or geographic regions; or
significant adverse effects on competition, employment, investment,
productivity, innovation, or on the ability of United States-based
enterprises to compete with foreign-based enterprises in domestic and
export markets.'' However, pursuant to the CRA, DEA has submitted a
copy of this final rule to both Houses of Congress and to the
Comptroller General.
List of Subjects in 21 CFR Part 1308
Administrative practice and procedure, Drug traffic control,
Reporting and recordkeeping requirements.
For the reasons set out above, 21 CFR part 1308 is amended as
follows:
PART 1308--SCHEDULES OF CONTROLLED SUBSTANCES
0
1. The authority citation for 21 CFR part 1308 continues to read as
follows:
Authority: 21 U.S.C. 811, 812, 871(b), 956(b), unless otherwise
noted.
0
2. In Sec. 1308.11:
0
a. Revise paragraphs (b)(22), (40), (56), and (59);
0
b. Add paragraph (b)(75);
0
c. Remove and reserve paragraphs (h)(23), and (h)(25) through (h)(28).
The revisions and addition read as follows:
Sec. 1308.11 Schedule I.
* * * * *
(b) * * *
(22) Cyclopentyl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9847
phenylcyclopentanecarboxamide)............................
* * * * * * *
(40) Isobutyryl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9827
phenylisobutyramide)......................................
* * * * * * *
(56) para-Chloroisobutyryl fentanyl (N-(4-chlorophenyl)-N- 9826
(1-phenethylpiperidin-4-yl)isobutyramide..................
[[Page 75235]]
* * * * * * *
(59) para-Methoxybutyryl fentanyl (N-(4-methoxyphenyl)-N-(1- 9837
phenethylpiperidin-4-yl)butyramide).......................
* * * * * * *
(75) Valeryl fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9840
phenylpentanamide)........................................
* * * * *
Timothy J. Shea,
Acting Administrator.
[FR Doc. 2020-22757 Filed 11-24-20; 8:45 am]
BILLING CODE 4410-09-P