Government-Owned Inventions; Availability for Licensing, 4571-4573 [2010-1680]
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mstockstill on DSKH9S0YB1PROD with NOTICES
Federal Register / Vol. 75, No. 18 / Thursday, January 28, 2010 / Notices
all of the images to perform a localized
analysis (corresponding X–Y pixels or
X–Y–Z voxels are analyzed across all
images) that identifies temporal
components within each sub-region.
Subsequently, within the sub-regions,
only those temporal components are
selected whose amplitude is above a
predetermined amplitude threshold.
The images are then reconstructed using
the sub-regions with reduced
components. A maximal-intensityprojection (MIP) is applied in the
temporal domain (tMIP) in order to
obtain a single image with reduced
noise (this can be done either at the subregion level or at the reconstructed
image level). The technology can be
applied to a broad spectrum of medical
imaging technologies such as MRI, XRay, CT and others.
Applications: Medical imaging and
diagnostics applied to MRI, X-Ray, CT
scans or other imaging modalities
including PET, SPECT, ultrasound or
optical.
Advantages: Enhancing signal-tonoise of medical imaging techniques.
Development Status:
• Proof of concept has been
demonstrated. Data is available.
• Need to acquire further data to
establish clinical utility of the method
and to further optimize the protocol.
Market:
• According to market research
reports the market for medical imaging
equipment industry in the United States
is approximately $9.0 billion dollars
now and has been growing by
approximately 7.6% annually.
• The United States market for
computed tomography (CT) scanning
systems is estimated to touch $3.6
billion by the end of 2009. The U.S.
accounts for over 50.0% of the
worldwide market.
• Worldwide MRI equipment market
is estimated to reach $5.5 billion by
2010, according to new report by Global
Industry Analysts, Inc. (https://www.
strategyr.com/Magnetic_Resonance_
Imaging_MRI_Equipment_Market_
Report.asp). In the United States the
market for such equipment is estimated
at $1.9 billion for 2008, as stated the
same report. The very high-field MRI
systems market in the United States is
projected to reach $968 million by the
year 2010. Very High-Field Systems also
represent the fastest growing segment,
as hospitals and clinics upgrade old
equipment with state-of-the-art systems.
• Enhancements in imaging
technologies to achieve better image
clarity, reliability and speed are being
constantly pursued by medical imaging
companies. Technologies that offer such
improvements therefore present
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excellent commercial potential. Thus
the subject invention which can be
applied in a broad spectrum of imaging
technologies offers such good
commercial potential.
Inventors: Han Wen and Vinay Pai
(NHLBI).
Relevant Articles:
1. Fish DA, Grochmalicki J, Pike ER.
Scanning singular-value-decomposition
method for restoration of images with
space-variant blur. J Opt Soc Am A,
13(3), pp. 464–469, March 1996.
2. Du X, Dunxu Y, Cuihua L, Jing L.
‘‘A novel approach to SVD-based image
filtering improvement,’’ International
Conference on Computer Science and
Software Engineering, vol 6, pp. 133–
136, 2008.
Patent Status: U.S. Provisional
Application No. 61/266,442 filed
December 3, 2009, entitled ‘‘Signal-toNoise Enhancement in Imaging
Applications Using a Time-Series of
Images’’ (HHS Reference No. E–292–
2009/0–US–01).
Related Technologies: Image
denoising techniques such as singular
value decomposition (SVD).
Licensing Status: Available for
licensing.
Licensing Contacts: Uri Reichman,
Ph.D., MBA; 301–435–4616;
UR7a@nih.gov; or John Stansberry,
Ph.D.; 301–435–5236;
stansbej@mail.nih.gov.
Collaborative Research Opportunity:
The National Heart, Lung, and Blood
Institute is seeking statements of
capability or interest from parties
interested in collaborative research to
implement the technology described
above on specific commercial platforms.
Please contact Denise Crooks, Ph.D. at
301–435–0103 or via e-mail at
crooksd@nhlbi.nih.gov for more
information.
Method for the Treatment of HIV/AIDS
Infection Using Acyclovir in Identified
Subjects
Description of Invention: The
invention provides the novel method to
treat HIV infections with acyclovir
which can be converted to acyclovir
triphosphate inside infected cells.
Acyclovir or acyclovir-related drugs
were previously approved for control of
herpesvirus replication with 20 years of
records of safe application. The subject
invention demonstrates that acyclovir
triphosphate can inhibit HIV–1 reverse
transcriptase as a potent suppressor of
HIV–1 replication in human lymphoid
tissues. In addition, the subject
invention may be attractive to potential
licensees, as there is little to no FDA
hurdle to overcome in the development
of the new formulations to use in this
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manner. Thus, the low cost and proven
safety of acyclovir may lead to a new
medicine for treating HIV–1 infections
and a prophylactic agent for preventing
HIV infections.
Applications: The treatment and
prevention of HIV infections.
Development Status: In vitro data
available.
Inventors: Leonid B. Margolis, Andrea
Lisco, Christophe Vanpouille, JeanCharles Grivel (NICHD).
Related Publications:
1. A Lisco et al. Acyclovir is activated
into a HIV–1 reverse transcriptase
inhibitor in herpesvirus-infected human
tissues. Cell Host Microbe. 2008 Sep
11;4(3):260–270. [PubMed: 18779052]
2. N Nagot et al. Reduction of HIV–
1 RNA levels with therapy to suppress
herpes simplex virus. New Engl J Med.
2007 Feb 22;356(8):790–799. [PubMed:
17314338]
Patent Status: PCT Application No.
PCT/US2008/010316 filed 30 Aug 2008,
which published as WO 2009/032244
on 12 Mar 2009 (HHS Reference No. E–
306–2007/0–PCT–02).
Licensing Status: Available for
licensing.
Licensing Contact: Sally Hu, Ph.D.;
301/435–5606; HuS@mail.nih.gov.
Collaborative Research Opportunity:
The Eunice Kennedy Shriver National
Institute of Child Health and Human
Development, Program in Physical
Biology, Section on Intracellular
Interactions, is seeking statements of
capability or interest from parties
interested in collaborative research to
further develop, evaluate, or
commercialize this technology. Please
contact Joseph Conrad, Ph.D., J.D. at
301–435–3107 or
jmconrad@mail.nih.gov for more
information.
Dated: January 21, 2010.
Richard U. Rodriguez,
Director, Division of Technology Development
and Transfer, Office of Technology Transfer,
National Institutes of Health.
[FR Doc. 2010–1669 Filed 1–27–10; 8:45 am]
BILLING CODE 4140–01–P
DEPARTMENT OF HEALTH AND
HUMAN SERVICES
National Institutes of Health
Government-Owned Inventions;
Availability for Licensing
AGENCY: National Institutes of Health,
Public Health Service, HHS.
ACTION: Notice.
SUMMARY: The inventions listed below
are owned by an agency of the U.S.
E:\FR\FM\28JAN1.SGM
28JAN1
4572
Federal Register / Vol. 75, No. 18 / Thursday, January 28, 2010 / Notices
mstockstill on DSKH9S0YB1PROD with NOTICES
Government and are available for
licensing in the U.S. in accordance with
35 U.S.C. 207 to achieve expeditious
commercialization of results of
federally-funded research and
development. Foreign patent
applications are filed on selected
inventions to extend market coverage
for companies and may also be available
for licensing.
ADDRESSES: Licensing information and
copies of the U.S. patent applications
listed below may be obtained by writing
to the indicated licensing contact at the
Office of Technology Transfer, National
Institutes of Health, 6011 Executive
Boulevard, Suite 325, Rockville,
Maryland 20852–3804; telephone: 301/
496–7057; fax: 301/402–0220. A signed
Confidential Disclosure Agreement will
be required to receive copies of the
patent applications.
Mouse Macula Densa Cell Line
Description of Invention: This
technology provides a clonally derived
macula densa cell line (MMDD1 cells)
that closely mimics the known
molecular expression pattern of native
macula densa (MD) cells. MMDD1 cells
are developed from SV–40 transgenic
mice using fluorescence-activated cell
sorting of renal tubular cells labeled
with segment-specific fluorescent
lectins. The MMDD1 cells of this
technology express COX–2, bNOS,
NKCC2, and ROMK, but not TammHorsfall protein, and show rapid 86Rb+
uptake that is inhibited by a reduction
in NaCl concentration and by
bumetanide or furosemide. These
MMDD1 cells provide a useful in vitro
model for the study of Macula Densa
function.
¨
Inventor: Jurgen B. Schnermann
(NIDDK).
Publication: T Yang, JM Park, L
Arend, Y Huang, R Topaloglu, A
Pasumarthy, H Praetorius, K Spring, JP
Briggs, J Schnermann. Low chloride
stimulation of prostaglandin E2 release
and cyclooxygenase-2 expression in a
mouse macula densa cell line. J Biol
Chem. 2000 Dec 1;275(48):37922–37929.
[PubMed: 10982805].
Patent Status: HHS Reference No. E–
234–2009/0—Research Tool. Patent
protection is not being pursued for this
technology.
Licensing Status: Available for
licensing under a Biological Materials
License Agreement.
Licensing Contact: Suryanarayana
(Sury) Vepa, Ph.D., J.D.; 301–435–5020;
vepas@mail.nih.gov.
Collaborative Research Opportunity:
The National Institute of Diabetes and
Digestive and Kidney Diseases Kidney
Disease Branch is seeking statements of
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17:16 Jan 27, 2010
Jkt 220001
capability or interest from parties
interested in collaborative research to
further develop, evaluate, or
commercialize the clonally derived
macula densa cell line (MMDD1 cells).
Please contact Cindy Fuchs at 301–451–
3636 for more information.
Novel Analogues of the Natural Product
Schweinfurthin With Specificity for
Tumors and Other Disease
Manifestations Associated With
Neurofibromatosis Type 1
Description of Invention: The global
anti-cancer market is forecast to reach
$40 billion by 2012. There remains a
significant unmet need for therapies to
treat neurofibromatosis type 1 (‘‘NF1’’), a
common genetic disease that afflicts 1 in
3500 people, and malignant tumors
carrying NF1 mutations, including
tumors of the central and peripheral
nervous systems.
Researchers at the National Cancer
Institute (‘‘NCI’’)-Frederick investigating
genetic influences on cancer
susceptibility of the nervous system
have synthesized novel analogues of
Schweinfurthin, a natural compound
first isolated from the tropical African
plant Macaranga schweinfurthii, to
which glioma and leukemia cell lines
show significant sensitivity. The
Schweinfurthin analogues also have
inhibitory activity against mouse and
human NF1 cancer cell lines. The
analogues have a novel mode of action
that appears to involve regulation of
cytoskeletal reorganization.
These inhibitors are likely to be
accepted in the marketplace because
their potent, selective activity and
unique specificity in mode of action
gives them a distinct advantage over the
mechanisms of other existing therapies.
Applications:
• Therapies for tumors associated
with NF1 (including brain and
peripheral nervous system tumors).
• Therapies for leukemia.
• Therapies for NF1 and associated
conditions.
Advantages:
• Utilizes proven small-molecule
technology.
• Specificity of mode of action may
reduce potential side-effects.
• Novel mode of action may limit
market competition.
Development Status: Pre-clinical.
Inventors: Karlyne Reilly et al. (NCI).
Relevant Publication: Turbyville et
al., ‘‘Schweinfurthin A Selectively
Inhibits Proliferation and Rho Signaling
in Glioma and Neurofibromatosis type 1
Tumor Cells in an NF1–GRD Dependent
Manner’’, submitted.
Patent Status: U.S. Patent Application
No. 61/174,338, filed 30 Apr 2009 (HHS
Reference No. E–183–2009/0–US–01).
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Licensing Status: Available for
licensing.
Licensing Contact: Patrick P. McCue,
Ph.D.; 301–435–5560;
mccuepat@mail.nih.gov.
Collaborative Research Opportunity:
The Genetic Modifiers of Tumorigenesis
Section at the National Cancer InstituteFrederick is seeking statements of
capability or interest from parties
interested in collaborative research to
further develop, evaluate, or
commercialize Schweinfurthins for the
treatment of Neurofibromatosis type 1.
Please contact John D. Hewes, Ph.D. at
301–435–3121 or hewesj@mail.nih.gov
for more information.
Detection of Autoantibodies for the
Diagnosis of Sjogren’s Syndrome
Description of Invention: This
invention provides a method for
diagnosing Sjogren’s syndrome in a
subject. In tests utilizing blood from
human volunteers, this method
demonstrated dramatically higher
accuracy (76%) in positively diagnosing
Sjogren’s syndrome than a standard,
currently available immunoassay (46%).
Briefly, this invention employs a
panel of mammalian-derived proteins
and protein fragments that are often
antigentic in individuals with Sjogren’s
syndrome in concert with a luciferase
immunoprecipitation system. In
contrast, most currently available
immunoassays for diagnosis of
rheumatological diseases include either
antigens from recombinant bacterial
expression systems or single antigens
from bovine sources. These
immunoassays are likely to fail to
present the sufficient variety of specific
human epitopes that are necessary for
high accuracy diagnoses of Sjogren’s
syndrome.
Applications:
• Diagnosis of Sjogren’s syndrome.
• A component of a panel of
diagnostic tests for patients with
autoimmune disease symptoms.
Advantages: Higher accuracy than
currently available diagnostics of
Sjogren’s syndrome.
Development Status: Early stage.
Initial clinical screens have been
completed.
Market: According to the Sjogren’s
Syndrome Foundation, Inc., it takes on
average seven years for a positive
Sjogren’s syndrome diagnosis as
symptoms of this syndrome mimic other
conditions and diseases. Up to four
million individuals in the United States
have Sjogren’s syndrome, and half of
currently diagnosed cases occur in
concert with other autoimmune disease
(https://www.sjogrens.org/home/aboutsjogrens-syndrome).
E:\FR\FM\28JAN1.SGM
28JAN1
Federal Register / Vol. 75, No. 18 / Thursday, January 28, 2010 / Notices
Inventors: Peter D. Burbelo and
Michael J. Iadarola (NIDCR).
Related Publications:
1. Burbelo PD, Leahy HP, Issa AT,
Groot S, Baraniuk JN, Nikolov NP, Illei
GG, Iadarola MJ. Sensitive and robust
luminescent profiling of anti-La and
other autoantibodies in Sjogren’s
syndrome. Autoimmunity. 2009
Sep;42(6):515–524. [PubMed: 19657778]
2. Burbelo PD, Ching KH, Issa AT,
Loftus CM, Li Y, Satoh M, Reeves WH,
Iadarola MJ. Rapid serological detection
of autoantibodies associated with
¨
Sjogren’s syndrome. J Transl Med. 2009
Sep 24;7:83. [PubMed: 19778440]
3. Burbelo PD, Ching KH, Klimavicz
CM, Iadarola MJ. Antibody profiling by
Luciferase Immunoprecipitation
Systems (LIPS). J Vis Exp. 2009 Oct
7;(32); pii: 1549; doi: 10.3791/1549.
[PubMed: 19812534]
Patent Status: U.S. Provisional
Application No. 61/224,649 filed 10 Jul
2009 (HHS Reference No. E–070–2009/
0–US–01).
Licensing Status: Available for
licensing.
Licensing Contact: Norbert Pontzer,
J.D., Ph.D.; 301–435–5502;
pontzern@mail.nih.gov.
Collaborative Research Opportunity:
The National Institute of Dental and
Craniofacial Research, Laboratory of
Sensory Biology, Neurobiology and Pain
Therapeutics Section, is seeking
statements of capability or interest from
parties interested in collaborative
research to further develop, evaluate, or
commercialize this technology. Please
contact David W. Bradley, Ph.D. at 301–
402–0540 or bradleyda@nidcr.nih.gov
for more information.
Dated: January 21, 2010.
Richard U. Rodriguez,
Director, Division of Technology Development
and Transfer, Office of Technology Transfer,
National Institutes of Health.
[FR Doc. 2010–1680 Filed 1–27–10; 8:45 am]
BILLING CODE 4140–01–P
DEPARTMENT OF HEALTH AND
HUMAN SERVICES
National Institutes of Health
mstockstill on DSKH9S0YB1PROD with NOTICES
Government-Owned Inventions;
Availability for Licensing
AGENCY: National Institutes of Health,
Public Health Service, HHS.
ACTION: Notice.
SUMMARY: The inventions listed below
are owned by an agency of the U.S.
Government and are available for
licensing in the U.S. in accordance with
35 U.S.C. 207 to achieve expeditious
VerDate Nov<24>2008
17:16 Jan 27, 2010
Jkt 220001
commercialization of results of
federally-funded research and
development. Foreign patent
applications are filed on selected
inventions to extend market coverage
for companies and may also be available
for licensing.
ADDRESSES: Licensing information and
copies of the U.S. patent applications
listed below may be obtained by writing
to the indicated licensing contact at the
Office of Technology Transfer, National
Institutes of Health, 6011 Executive
Boulevard, Suite 325, Rockville,
Maryland 20852–3804; telephone:
301/496–7057; fax: 301/402–0220. A
signed Confidential Disclosure
Agreement will be required to receive
copies of the patent applications.
Nitric Oxide-Based Therapeutics for
Lung Cancer
Description of Invention: JS–36–25, a
diazeniumdiolate prodrug, is available
for licensing and development of
treatments for lung cancer. The
inventors have demonstrated a potent
tumoristatic activity of JS–36–25 in both
lung cancer cells in vitro and as
xenografts in mice. JS–36–25 treatment
led to 85% reduction of tumor growth
in vivo. The tumoristatic potency of the
compound correlated well with the
level of endogenous reactive oxygen
species (ROS) in the cancer cells. Thus,
in addition to potent tumoristatic
activity when administered alone, this
compound is predicted to have a strong
synergy with therapeutics that act
through generation of ROS, such as
bortezomib, doxorubicin, as well as
high-energy radiation.
Applications: Development of lung
cancer treatments.
Development Status: Pre-clinical.
Market: There are over 160,000 new
cases of lung cancer every year in the
United States alone.
Inventors: Anna E. Maciag et al. (NCI).
Patent Status: U.S. Provisional
Application No. 61/261,175 filed 13
November 2009 (HHS Reference No.
E–025–2010/0–US–01).
Licensing Status: Available for
licensing.
Licensing Contact: Steve Standley,
Ph.D.; 301–435–4074;
sstand@od.nih.gov.
T-Cell-Specific Gfi-1 Knockout Mouse
Description of Invention: This is a
mouse model available to study T-cell
differentiation. Growth factor
independent 1 (GFi-1) is a
transcriptional repressor that is
transiently induced during T-cell
activation. This knockout mouse line is
a GFi-1[flox/flox] introduced into a
mouse Cre controlled by a CD4
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4573
promoter, which allows selective
removal of GFi-1 exclusively in T-cells.
It has thus-far been used to demonstrate
that GFi-1 plays a critical role in
enhancing Th2 cell expansion and
repressing induction of Th17 and
CD103+ iTreg cells.
Applications: Tool for studying T-cell
proliferation and differentiation.
Inventors: Jinfang Zhu and William E.
Paul (NIAID).
Related Publication: J Zhu, TS
Davidson, G Wei, D Jankovic, K Cui, DE
Schones, L Guo, K Zhao, EM Shevach,
WE Paul. Down-regulation of Gfi-1
expression by TGF-beta is important for
differentiation of Th17 and CD103+
inducible regulatory T cells. J Exp Med.
2009 Feb 16;206(2):329–341. [PubMed:
19188499].
Patent Status: HHS Reference No.
E–242–2009/0—Research Tool. Patent
protection is not being pursued for this
technology.
Licensing Status: This technology is
available as a research tool under a
Biological Materials License.
Licensing Contact: Steve Standley,
Ph.D.; 301–435–4074;
sstand@od.noh.gov.
Dated: January 21, 2010.
Richard U. Rodriguez,
Director, Division of Technology Development
and Transfer, Office of Technology Transfer,
National Institutes of Health.
[FR Doc. 2010–1668 Filed 1–27–10; 8:45 am]
BILLING CODE 4140–01–P
DEPARTMENT OF HEALTH AND
HUMAN SERVICES
National Institutes of Health
Government-Owned Inventions;
Availability for Licensing
AGENCY: National Institutes of Health,
Public Health Service, HHS.
ACTION: Notice.
SUMMARY: The inventions listed below
are owned by an agency of the U.S.
Government and are available for
licensing in the U.S. in accordance with
35 U.S.C. 207 to achieve expeditious
commercialization of results of
Federally funded research and
development. Foreign patent
applications are filed on selected
inventions to extend market coverage
for companies and may also be available
for licensing.
ADDRESSES: Licensing information and
copies of the U.S. patent applications
listed below may be obtained by writing
to the indicated licensing contact at the
Office of Technology Transfer, National
Institutes of Health, 6011 Executive
E:\FR\FM\28JAN1.SGM
28JAN1
Agencies
[Federal Register Volume 75, Number 18 (Thursday, January 28, 2010)]
[Notices]
[Pages 4571-4573]
From the Federal Register Online via the Government Printing Office [www.gpo.gov]
[FR Doc No: 2010-1680]
-----------------------------------------------------------------------
DEPARTMENT OF HEALTH AND HUMAN SERVICES
National Institutes of Health
Government-Owned Inventions; Availability for Licensing
AGENCY: National Institutes of Health, Public Health Service, HHS.
ACTION: Notice.
-----------------------------------------------------------------------
SUMMARY: The inventions listed below are owned by an agency of the U.S.
[[Page 4572]]
Government and are available for licensing in the U.S. in accordance
with 35 U.S.C. 207 to achieve expeditious commercialization of results
of federally-funded research and development. Foreign patent
applications are filed on selected inventions to extend market coverage
for companies and may also be available for licensing.
ADDRESSES: Licensing information and copies of the U.S. patent
applications listed below may be obtained by writing to the indicated
licensing contact at the Office of Technology Transfer, National
Institutes of Health, 6011 Executive Boulevard, Suite 325, Rockville,
Maryland 20852-3804; telephone: 301/496-7057; fax: 301/402-0220. A
signed Confidential Disclosure Agreement will be required to receive
copies of the patent applications.
Mouse Macula Densa Cell Line
Description of Invention: This technology provides a clonally
derived macula densa cell line (MMDD1 cells) that closely mimics the
known molecular expression pattern of native macula densa (MD) cells.
MMDD1 cells are developed from SV-40 transgenic mice using
fluorescence-activated cell sorting of renal tubular cells labeled with
segment-specific fluorescent lectins. The MMDD1 cells of this
technology express COX-2, bNOS, NKCC2, and ROMK, but not Tamm-Horsfall
protein, and show rapid 86Rb+ uptake that is inhibited by a reduction
in NaCl concentration and by bumetanide or furosemide. These MMDD1
cells provide a useful in vitro model for the study of Macula Densa
function.
Inventor: J[uuml]rgen B. Schnermann (NIDDK).
Publication: T Yang, JM Park, L Arend, Y Huang, R Topaloglu, A
Pasumarthy, H Praetorius, K Spring, JP Briggs, J Schnermann. Low
chloride stimulation of prostaglandin E2 release and cyclooxygenase-2
expression in a mouse macula densa cell line. J Biol Chem. 2000 Dec
1;275(48):37922-37929. [PubMed: 10982805].
Patent Status: HHS Reference No. E-234-2009/0--Research Tool.
Patent protection is not being pursued for this technology.
Licensing Status: Available for licensing under a Biological
Materials License Agreement.
Licensing Contact: Suryanarayana (Sury) Vepa, Ph.D., J.D.; 301-435-
5020; vepas@mail.nih.gov.
Collaborative Research Opportunity: The National Institute of
Diabetes and Digestive and Kidney Diseases Kidney Disease Branch is
seeking statements of capability or interest from parties interested in
collaborative research to further develop, evaluate, or commercialize
the clonally derived macula densa cell line (MMDD1 cells). Please
contact Cindy Fuchs at 301-451-3636 for more information.
Novel Analogues of the Natural Product Schweinfurthin With Specificity
for Tumors and Other Disease Manifestations Associated With
Neurofibromatosis Type 1
Description of Invention: The global anti-cancer market is forecast
to reach $40 billion by 2012. There remains a significant unmet need
for therapies to treat neurofibromatosis type 1 (``NF1''), a common
genetic disease that afflicts 1 in 3500 people, and malignant tumors
carrying NF1 mutations, including tumors of the central and peripheral
nervous systems.
Researchers at the National Cancer Institute (``NCI'')-Frederick
investigating genetic influences on cancer susceptibility of the
nervous system have synthesized novel analogues of Schweinfurthin, a
natural compound first isolated from the tropical African plant
Macaranga schweinfurthii, to which glioma and leukemia cell lines show
significant sensitivity. The Schweinfurthin analogues also have
inhibitory activity against mouse and human NF1 cancer cell lines. The
analogues have a novel mode of action that appears to involve
regulation of cytoskeletal reorganization.
These inhibitors are likely to be accepted in the marketplace
because their potent, selective activity and unique specificity in mode
of action gives them a distinct advantage over the mechanisms of other
existing therapies.
Applications:
Therapies for tumors associated with NF1 (including brain
and peripheral nervous system tumors).
Therapies for leukemia.
Therapies for NF1 and associated conditions.
Advantages:
Utilizes proven small-molecule technology.
Specificity of mode of action may reduce potential side-
effects.
Novel mode of action may limit market competition.
Development Status: Pre-clinical.
Inventors: Karlyne Reilly et al. (NCI).
Relevant Publication: Turbyville et al., ``Schweinfurthin A
Selectively Inhibits Proliferation and Rho Signaling in Glioma and
Neurofibromatosis type 1 Tumor Cells in an NF1-GRD Dependent Manner'',
submitted.
Patent Status: U.S. Patent Application No. 61/174,338, filed 30 Apr
2009 (HHS Reference No. E-183-2009/0-US-01).
Licensing Status: Available for licensing.
Licensing Contact: Patrick P. McCue, Ph.D.; 301-435-5560;
mccuepat@mail.nih.gov.
Collaborative Research Opportunity: The Genetic Modifiers of
Tumorigenesis Section at the National Cancer Institute-Frederick is
seeking statements of capability or interest from parties interested in
collaborative research to further develop, evaluate, or commercialize
Schweinfurthins for the treatment of Neurofibromatosis type 1. Please
contact John D. Hewes, Ph.D. at 301-435-3121 or hewesj@mail.nih.gov for
more information.
Detection of Autoantibodies for the Diagnosis of Sjogren's Syndrome
Description of Invention: This invention provides a method for
diagnosing Sjogren's syndrome in a subject. In tests utilizing blood
from human volunteers, this method demonstrated dramatically higher
accuracy (76%) in positively diagnosing Sjogren's syndrome than a
standard, currently available immunoassay (46%).
Briefly, this invention employs a panel of mammalian-derived
proteins and protein fragments that are often antigentic in individuals
with Sjogren's syndrome in concert with a luciferase
immunoprecipitation system. In contrast, most currently available
immunoassays for diagnosis of rheumatological diseases include either
antigens from recombinant bacterial expression systems or single
antigens from bovine sources. These immunoassays are likely to fail to
present the sufficient variety of specific human epitopes that are
necessary for high accuracy diagnoses of Sjogren's syndrome.
Applications:
Diagnosis of Sjogren's syndrome.
A component of a panel of diagnostic tests for patients
with autoimmune disease symptoms.
Advantages: Higher accuracy than currently available diagnostics of
Sjogren's syndrome.
Development Status: Early stage. Initial clinical screens have been
completed.
Market: According to the Sjogren's Syndrome Foundation, Inc., it
takes on average seven years for a positive Sjogren's syndrome
diagnosis as symptoms of this syndrome mimic other conditions and
diseases. Up to four million individuals in the United States have
Sjogren's syndrome, and half of currently diagnosed cases occur in
concert with other autoimmune disease (https://www.sjogrens.org/home/about-sjogrens-syndrome).
[[Page 4573]]
Inventors: Peter D. Burbelo and Michael J. Iadarola (NIDCR).
Related Publications:
1. Burbelo PD, Leahy HP, Issa AT, Groot S, Baraniuk JN, Nikolov NP,
Illei GG, Iadarola MJ. Sensitive and robust luminescent profiling of
anti-La and other autoantibodies in Sjogren's syndrome. Autoimmunity.
2009 Sep;42(6):515-524. [PubMed: 19657778]
2. Burbelo PD, Ching KH, Issa AT, Loftus CM, Li Y, Satoh M, Reeves
WH, Iadarola MJ. Rapid serological detection of autoantibodies
associated with Sj[ouml]gren's syndrome. J Transl Med. 2009 Sep
24;7:83. [PubMed: 19778440]
3. Burbelo PD, Ching KH, Klimavicz CM, Iadarola MJ. Antibody
profiling by Luciferase Immunoprecipitation Systems (LIPS). J Vis Exp.
2009 Oct 7;(32); pii: 1549; doi: 10.3791/1549. [PubMed: 19812534]
Patent Status: U.S. Provisional Application No. 61/224,649 filed 10
Jul 2009 (HHS Reference No. E-070-2009/0-US-01).
Licensing Status: Available for licensing.
Licensing Contact: Norbert Pontzer, J.D., Ph.D.; 301-435-5502;
pontzern@mail.nih.gov.
Collaborative Research Opportunity: The National Institute of
Dental and Craniofacial Research, Laboratory of Sensory Biology,
Neurobiology and Pain Therapeutics Section, is seeking statements of
capability or interest from parties interested in collaborative
research to further develop, evaluate, or commercialize this
technology. Please contact David W. Bradley, Ph.D. at 301-402-0540 or
bradleyda@nidcr.nih.gov for more information.
Dated: January 21, 2010.
Richard U. Rodriguez,
Director, Division of Technology Development and Transfer, Office of
Technology Transfer, National Institutes of Health.
[FR Doc. 2010-1680 Filed 1-27-10; 8:45 am]
BILLING CODE 4140-01-P